CAS No. : 1616391-87-7

(Synonyms: EPZ015866; GSK3203591)

Price and Availability of CAS No. : 1616391-87-7
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10mg $216 In-stock
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100mg $1140 In-stock
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Cat. No. : HY-100235
M.Wt: 380.48
Formula: C22H28N4O2
Purity: >98 %
Solubility: DMSO : ≥ 135 mg/mL (354.81 mM)
Introduction of 1616391-87-7 :

GSK591 (EPZ015866) is a potent and selective inhibitor of protein methyltransferase 5 (PRMT5) with an IC50 of 4 nM[1]. IC50 & Target: IC50: 4 nM (PRMT5)[1] In Vitro: GSK591 (5 μM; MCF7, T47D, and MCF10A cells) treatment suppresses breast cancer stem cells (BCSCs) proliferation and self-renewal. GSK591 reduces BCSCs numbers in vitro[2].

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