U93631


CAS No. : 152273-12-6

152273-12-6
Price and Availability of CAS No. : 152273-12-6
Size Price Stock
5mg $50 In-stock
10mg $80 In-stock
25mg $160 In-stock
50mg $250 In-stock
100mg $900 In-stock
200 mg Get quote
500 mg Get quote
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Cat. No. : HY-100686
M.Wt: 299.37
Formula: C17H21N3O2
Purity: >98 %
Solubility: DMSO : ≥ 34 mg/mL (113.57 mM)
Introduction of 152273-12-6 :

U93631 is a GABAA receptor ligand of novel chemical structure with IC50 of 100 nM,and has been shown to induce a rapid, time-dependent decay of GABA-induced whole-cell Cl-currents in recombinant GABAA receptors. target: GABAA receptor IC 50: GABAA receptor[1] In vitro: In the presence of U93631 at 5 UM, the peak amplitude decreased as a function of GABA concentration, with the half-maximal inhibitory concentration being approximately 100 nM, which is close to the Kd for the high affinity GABA site(85 nM). It appears that the drug interacts with GABA-bound receptors (at least monoliganded) and accelerates receptor desensitization, rather than acting as an open channel blocker. [1]

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