Size | Price | Stock |
---|---|---|
1mg | $30 | In-stock |
5mg | $65 | In-stock |
10mg | $111 | In-stock |
25mg | $221 | In-stock |
50 mg | Get quote | |
100 mg | Get quote | |
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Cat. No. : | HY-100398 |
M.Wt: | 446.50 |
Formula: | C24H26N6O3 |
Purity: | >98 % |
Solubility: | DMSO : 10 mg/mL (22.40 mM; Need ultrasonic) |
PF-04979064 is a potent and selective PI3K/mTOR dual kinase inhibitor with Kis of 0.13 nM and 1.42 nM for PI3Kα and mTOR, respectively. IC50 & Target:Ki: 0.13 nM (PI3Kα), 1.42 nM (mTOR)[1] In Vitro: PF-04979064 is tested against human class I PI3K isoforms PI3Kα, PI3Kγ, and PI3Kδ, with PI3Kα Ki of 0.13 nM, PI3Kγ Ki of 0.111 nM, and PI3Kδ Ki of 0.122 nM[1]. In Vivo: PF-04979064 is progressed to rat in vivo PK studies and exhibits robust PK profile: Vdss=5.23 L/kg, Cl=19.3 mL/min/kg, T1/2=1.85 h, and F%=61%[1].
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