Size | Price | Stock |
---|---|---|
5mg | $150 | In-stock |
10mg | $250 | In-stock |
25mg | $490 | In-stock |
50mg | $780 | In-stock |
100 mg | Get quote | |
200 mg | Get quote | |
We match the lowest price on market. |
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
Cat. No. : | HY-100064 |
M.Wt: | 432.88 |
Formula: | C21H22ClFN4O3 |
Purity: | >98 % |
Solubility: | 10 mM in DMSO |
O-Desmethyl gefitinib is an active metabolite of Gefitinib in human plasma. The formation of O-desmethyl gefitinib is dependent on CYP2D6 activity. O-desmethyl gefitinib inhibits EGFR with an IC50 of 36 nM in subcellular assays[1][2]. IC50 & Target:IC50: 36 nM (EGFR)[2]
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information
Your information is safe with us.