Pentiapine
CAS No. : 81382-51-6
(Synonyms: CGS 10746)
| Size | Price | Stock |
|---|---|---|
| 1mg | $751 | In-stock |
| 5mg | $1202 | In-stock |
| 10mg | $1923 | In-stock |
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| 100 mg | Get quote | |
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| Cat. No. : | HY-100143 |
| M.Wt: | 299.39 |
| Formula: | C15H17N5S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Pentiapine (CGS 10746) is a dopamine release inhibitor without binding to synaptic dopamine receptor sites[1][2]. IC50 & Target: Dopamine receptor[1] In Vivo: Pentiapine is a novel dopamine release inhibitor.The results show that Pentiapine dose-dependently reduces motor activity of mice. Moreover, Pentiapine dose-dependently reduces morphine-induced hyperactivity. Newman-Keuls post-hoc comparisons indicate that the group receiving morphine plus saline presents more activity than the groups receiving morphine plus 2 (P<0.05), 4, 8, 16, 24 and 32 (P<0.01) mg/kg of Pentiapine. Moreover, the groups receiving morphine plus 0.5, 1 and 2 mg/kg of Pentiapine present more activity than the groups receiving morphine plus 4, 8, 16, 24 and 32 mg/kg of Pentiapine (P<0.01)[1]. 30 mg/kg dose of Pentiapine completely blocks the methylenedioxymethamphetamine (MDMA) conditioned place preference (CPP) and also blocks the establishment of a cocaine CPP[2].
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