Vorapaxar
CAS No. : 618385-01-6
(Synonyms: SCH 530348)
| Size | Price | Stock |
|---|---|---|
| 1mg | $88 | In-stock |
| 5mg | $185 | In-stock |
| 10mg | $280 | In-stock |
| 25mg | $500 | In-stock |
| 50mg | $750 | In-stock |
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| Cat. No. : | HY-10119 |
| M.Wt: | 492.58 |
| Formula: | C29H33FN2O4 |
| Purity: | >98 % |
| Solubility: | DMSO : 25 mg/mL (50.75 mM; Need ultrasonic) |
Vorapaxar (SCH 530348), an antiplatelet agent, is a selective, orally active, and competitive thrombin receptor protease-activated receptor (PAR-1) antagonist (Ki=8.1 nM). Vorapaxar (SCH 530348) inhibits thrombin receptor-activating peptide (TRAP)-induced platelet aggregation in a dose-dependent manner[1]. IC50 & Target: Ki: 8.1 nM (PAR-1)[1] In Vitro: Vorapaxar (SCH 530348) shows potent inhibition of thrombin-induced platelet aggregation with an IC50 of 47 nM and haTRAP-induced platelet aggregation with an IC50 of 25 nM. Vorapaxar (SCH 530348) inhibits thrombininduced calcium transient in human coronary artery smooth muscle cells (HCASMC) with a Ki of 1.1 nM. It also inhibits thrombin-stimulated thymidine incorporation in HCASMC with a Ki of 13 nM[1].
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