Size | Price | Stock |
---|---|---|
5mg | $120 | In-stock |
10mg | $190 | In-stock |
25mg | $350 | In-stock |
50mg | $550 | In-stock |
100mg | $950 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-100113 |
M.Wt: | 475.62 |
Formula: | C23H29N3O4S2 |
Purity: | >98 % |
Solubility: | DMSO : 100 mg/mL (210.25 mM; Need ultrasonic) |
AT2 receptor agonist C21 is a druglike selective angiotensin II AT2 receptor agonist with Ki values of 0.4 nM and >10 µM for the AT2 receptor and AT1 receptor, respectively[1]. IC50 & Target:Ki: 0.4 nM (AT2) and >10 µM (AT1)[1] In Vivo: AT2 receptor agonist C21, with a bioavailability of 20-30% after oral administration and a half-life estimated to 4 h in rat, induces outgrowth of neurite cells, stimulates p42/p44mapk, enhances in vivo duodenal alkaline secretion in Sprague-Dawley rats, and lowers the mean arterial blood pressure in anesthetized, spontaneously hypertensive rats[1].
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