Size | Price | Stock |
---|---|---|
5mg | $300 | In-stock |
10mg | $450 | In-stock |
25mg | $950 | In-stock |
50mg | $1500 | In-stock |
100mg | $2400 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-100170 |
M.Wt: | 480.62 |
Formula: | C23H36N4O5S |
Purity: | >98 % |
Solubility: | 10 mM in DMSO |
5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. IC50 & Target:pKI: 9.6 (5-HT4 receptor)[1] In Vitro: 5-HT4 antagonist 1 (compound 6b) is a 5-HT4 receptor antagonist with a pKi of 9.6. In Vivo: 5-HT4 antagonist 1 (compound 6b) demonstrates good exposure and prolongs t1/2 in other species, including the mouse (t1/2 7 h), rat (t1/2 12 h) and mini-pig (t1/2 21 h). In Phase I clinical trial, it is found that 5-HT4 antagonist 1 has good oral bioavailability with a steady state plasma t1/2 of >100 h[1].
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