J-104132


CAS No. : 198279-45-7

(Synonyms: L 753037)

198279-45-7
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Cat. No. : HY-10383
M.Wt: 531.60
Formula: C31H33NO7
Purity: >98 %
Solubility: DMSO
Introduction of 198279-45-7 :

J-104132 is a potent, orally active ETA/ETB receptor antagonist, with Kis of 0.034 nM and 0.104 nM for cloned human ETA and ETB receptors expressed in CHO cells. IC50 & Target: Ki: 0.034 nM (human ETA receptor, CHO cell), 0.104 nM (human ETB receptor, CHO cell)[1] In Vitro: J-104132 is a potent, orally active mixed ETA/ETB receptor antagonist, with Kis of 0.034 nM and 0.104 nM for cloned human ETA and ETB receptors expressed in CHO cells. J-104132 also shows Ki of 0.350 ± 0.158 nM for ETA receptor in human uterus and 0.343 ± 0.146 nM for ETB receptor in human hippocampus[1].

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