(1R,2R)-2-PCCA(hydrochloride)
CAS No. : 1609563-71-4
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| Cat. No. : | HY-100013A1 |
| M.Wt: | 528.56 |
| Formula: | C30H39Cl2N3O |
| Purity: | >98 % |
| Storage: | at 20℃ 2 years |
| Solubility: | DMSO : 50 mg/mL (94.60 mM; Need ultrasonic) |
(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. IC50 & Target: EC50: 3 nM (GPR88 receptor)[1], 603 nM (GPR88 receptor, in GPR88-22F cells)[2] In Vitro: (1R,2R)-2-PCCA (Example 3) is a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay[1][2]. (1R,2R)-2-PCCA inhibits GPR88-mediated cAMP production through a Gαi-coupled pathway, with an EC50 of 56 nM in HEK293 cells stably expressing the human GPR88 receptor and the GloSensor-22F cAMP construct[2].
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