Size | Price | Stock |
---|---|---|
5mg | $50 | In-stock |
10mg | $80 | In-stock |
25mg | $150 | In-stock |
50mg | $250 | In-stock |
100mg | $400 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-100552 |
M.Wt: | 262.74 |
Formula: | C13H15ClN4 |
Purity: | >98 % |
Solubility: | 10 mM in DMSO |
VUF10166 is a potent and high-affinity 5-HT3 receptor antagonist, with Ki values of 0.04 nM (5-HT3A) and 22 nM (5-HT3AB). VUF10166 inhibits 5-HT-induced responses at 5-HT3A and 5-HT3AB receptors at nanomolar concentrations. At 5-HT3 receptor, VUF10166 at higher concentrations also acts as a partial agonist, with an EC50 of 5.2 μM[1]. IC50 & Target: IC50: 40 nM (5-HT3AB); Ki: 0.04 nM (5-HT3A), 22 nM (5-HT3AB)[1]
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