Size | Price | Stock |
---|---|---|
5mg | $820 | In-stock |
10mg | $1300 | In-stock |
25mg | $2600 | In-stock |
50mg | $4160 | In-stock |
100mg | $6650 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-103493 |
M.Wt: | 458.36 |
Formula: | C19H18F4N4O5 |
Purity: | >98 % |
Solubility: | DMSO : 7.5 mg/mL (16.36 mM; ultrasonic and warming and heat to 60°C) |
TAK-915 is a potent, selective, brain-penetrant and orally active phosphodiesterase 2A (PDE2A) inhibitor with an IC50 of 0.61 nM. TAK-915 is >4100-fold more selectivity for PDE2A than PDE1A. TAK-915 has the potential for neuropsychiatric and neurodegenerative disorders treatment[1][2].
In Vivo: TAK-915 (3 mg/kg; oral administration; daily; for 4 days; male F344 rats) treatment significantly reduces escape latency in aged rats in the Morris water maze task[2].
TAK-915 (1, 3, and 10 mg/kg, p.o.) dose-dependently attenuates the non-selective muscarinic antagonist scopolamine-induced memory deficits in rats[2].
Oral dosing of TAK-915 (compound 36) (3 or 10 mg/kg) in mice produces a dose-dependent increase in 3',5'-cyclic guanosine monophosphate (cGMP) levels, with significant cGMP increases observed at a dose of 10 mg/kg[1].
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