Size | Price | Stock |
---|---|---|
2mg | $106 | In-stock |
5mg | $132 | In-stock |
10mg | $198 | In-stock |
25mg | $330 | In-stock |
50mg | $594 | In-stock |
100mg | $990 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-100015 |
M.Wt: | 459.47 |
Formula: | C22H19F2N3O4S |
Purity: | >98 % |
Solubility: | DMSO : 100 mg/mL (217.64 mM; Need ultrasonic) |
Mivebresib (ABBV-075) is a potent and orally active bromodomain and extraterminal domain (BET) bromodomain inhibitor. Mivebresib binds to BRD4 with a Ki of 1.5 nM[1]. IC50 & Target: IC50: 1.5 nM (BRD4)[1] In Vitro: Mivebresib inhibit DHT-stimulated transcription of AR target genes without significant effect on AR protein expression. In addition to blocking the transcription activation downstream of AR, Mivebresib is also a potent inhibitor of MYC and the TMPRSS2-ETS fusion proteins[1].
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