Xanomeline (oxalate)
CAS No. : 141064-23-5
(Synonyms: LY246708 (oxalate))
| Size | Price | Stock |
|---|---|---|
| 5mg | $70 | In-stock |
| 10mg | $110 | In-stock |
| 50mg | $350 | In-stock |
| 100mg | $560 | In-stock |
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| Cat. No. : | HY-13410 |
| M.Wt: | 371.45 |
| Formula: | C16H25N3O5S |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (134.61 mM; Need ultrasonic) |
Xanomeline oxalate (LY246708 oxalate) is a potent and selective muscarinic receptor agonist (SMRA) and stimulates phosphoinositide hydrolysis in vivo. Xanomeline oxalate can be used for the research of Alzheimer’s disease[1].
IC50 & Target: muscarinic receptor[1]
In Vitro: Xanomeline stimulates phosphoinositide (PI) hydrolysis in the A9 L m1 cells[1].
Xanomeline inhibits [3H]-pirenzepine ([3H]-PZ) and [3H]-oxotremorine-M ([3H]-OXO-M) binding to rat brain with Kis of 7 and 3 nM, respectively[1].
In Vivo: Xanomeline robustly stimulates in vivo PI hydrolysis and the effect is blocked by muscarinic antagonists, demonstrating mediation by muscarinic receptors. In mice the ED100 for Xanomeline-induced stimulation of [3H]-IP accumulation is 54 μmole/kg in hippocampus. And in rats the ED100 for Xanomeline-induced stimulation of [3H]-IP accumulation is 8.1 μmole/kg in hippocampus[1].
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