(1R,2R)-2-PCCA
CAS No. : 1287205-42-8
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| Cat. No. : | HY-100013A |
| M.Wt: | 455.63 |
| Formula: | C30H37N3O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
(1R,2R)-2-PCCA is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. IC50 & Target: EC50: 3 nM (GPR88 receptor)[1], 603 nM (GPR88 receptor, in GPR88-22F cells)[2] In Vitro: (1R,2R)-2-PCCA (Example 3) is a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay[1][2]. (1R,2R)-2-PCCA inhibits GPR88-mediated cAMP production through a Gαi-coupled pathway, with an EC50 of 56 nM in HEK293 cells stably expressing the human GPR88 receptor and the GloSensor-22F cAMP construct[3].
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