Calpeptin
CAS No. : 117591-20-5
| Size | Price | Stock |
|---|---|---|
| 5mg | $66 | In-stock |
| 10mg | $95 | In-stock |
| 25mg | $198 | In-stock |
| 50mg | $280 | In-stock |
| 100mg | $450 | In-stock |
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| Cat. No. : | HY-100223 |
| M.Wt: | 362.46 |
| Formula: | C20H30N2O4 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (275.89 mM; Need ultrasonic) |
Calpeptin is a potent, cell penetrating calpain inhibitor, with an ID50 of 40 nM for Calpain I in human platelets[1]. Calpeptin is also an inhibitor of cathepsin K[2].
IC50 & Target: ID50: 40 nM (Calpain I in human platelets)[1].
Cthepsin K[2]
In Vitro: Calpeptin (0-100 nM, 24 hours) treatment suppresses the proliferation of both WI38 VA13 and IMR90 cells in a dose-dependent manner. Calpeptin (1000 pg/ml, 24 hours) inhibits IL-6-induced cell proliferation of lung fibroblasts[3].
In Vivo: Calpeptin with Bleo (0.04 mg/mouse, i.p., 3 times weekly, 28 days) administration significantly inhibits the collagen deposition and increases of calpain activity in the NSC-125066 treated mouse lung tissues[3].
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