Size | Price | Stock |
---|---|---|
5mg | $346 | In-stock |
10mg | $554 | In-stock |
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100 mg | Get quote | |
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Cat. No. : | HY-103461 |
M.Wt: | 397.38 |
Formula: | C19H17F2N7O |
Purity: | >98 % |
Solubility: | 10 mM in DMSO |
FAAH-IN-6 (compound 21d) is a potent, orally active and cross the blood-brain barrier fatty acid amide hydrolase (FAAH) inhibitor with IC50s of 0.72, 0.28 nM for hFAAH, rFAAH, respectively. FAAH-IN-6 shows dose-dependent analgesic efficacy in animal models of both neuropathic and inflammatory pain[1].
IC50 & Target: IC50: 0.72 nM (hFAAH); 0.28 nM (rFAAH)[1]
In Vivo: FAAH-IN-6 (compound 21d) (1-10 mg/kg; p.o.) shows significantly ameliorates tactile allodynia in a dose-dependent fashion in SNI-induced neuropathic pain rats model[1].
FAAH-IN-6 (3-10 mg/kg; p.o.) shows significantly ameliorates tactile allodynia of the ipsilateral hind paw in CFA-induced inflammatory pain model[1].
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